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信号通路, 信号转导, Cell Signaling

20,000多种特异性抑制剂、激动剂作用于表观遗传学、PI3K/Akt/mTOR、凋亡、MAPK、Wnt等20多个信号通路的375个靶点蛋白,覆盖癌症、神经科学、免疫学等热门疾病研究领域。BSZH北实纵横科学公司的50多种活性化合物库,包含10,000多种具有生物活性的小分子化合物,可用于高通量筛选 (HTS)和高内涵筛选 (HCS),是进行新药筛选和新适应症发现等研究的专业工具。

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GRN-529,≥97% (HPLC)

PZ0293
别名:[4-(二氟甲氧基)-3-[2-(2-吡啶基)乙炔基]苯基](5,7-二氢-6H-吡咯并[3,4-b]吡啶-6-基)-甲酮;[4-(Difluoromethoxy)-3-[2-(2-pyridinyl)ethynyl]phenyl](5,7-dihydro-6H-pyrrolo[3,4-b]pyridin-6-yl)-methanone

Empirical Formula (Hill Notation): C22H15F2N3O2 CAS号: 1253291-12-1 分子量: 391.37 MDL编号: MFCD28160551 PubChem化学物质编号: 329823817
¥5,760.00

ILS-920,≥98% (HPLC)

PZ0329
ILS920;Empirical Formula (Hill Notation): C57H86N2O14 CAS号: 892494-07-4 分子量: 1023.30 NACRES: NA.77
¥1,591.58

ISOX-DUAL,≥98% (HPLC)

PZ0331
别名:3-(4-(2-(5-(3,5-二甲基异恶唑-4-基)-1-(2-吗啉乙基)-1H-苯并[d]咪唑-2-基)乙基)苯氧基)-N, N-二甲基丙-1-胺;3-(4-(2-(5-(3,5-dimethylisoxazol-4-yl)-1-(2-morpholinoethyl)-1H-benzo[d]imidazol-2-yl)ethyl)phenoxy)-N,N-dimethylpropan-1-amine

Empirical Formula (Hill Notation): C31H41N5O3 分子量: 531.69 PubChem化学物质编号: 329823842 NACRES: NA.77
¥1,591.58

ISOX-INACT,≥98% (HPLC)

PZ0332
别名:4-(2-(5-(3,5-二甲基异恶唑-4-基)-2-(4-甲氧基苯乙基)-4,6-二甲基-1H苯并[d]咪唑-1-基)乙基)吗啉;4-(2-(5-(3,5-Dimethylisoxazol-4-yl)-2-(4-methoxyphenethyl)-4,6-dimethyl-1Hbenzo[d]imidazol-1-yl)ethyl)morpholine

Empirical Formula (Hill Notation): C29H36N4O3 分子量: 488.62 PubChem化学物质编号: 329823843 NACRES: NA.77
¥1,591.58

那法瑞林醋酸盐水合物,Nafarelin acetate salt hydrate;≥95% (HPLC), solid

N7662
别名:那法瑞林乙酸盐水合物;5-氧代-L-脯氨酰-L-组氨酸基-L-色叶基-L-丝氨酸-L-酪酰基-3-(2-萘基)-D-丙氨酰基-L-亮氨酸-L-精氨酸基-L-脯氨酰甘氨酰胺乙酸盐水合物;5-Oxo-L-prolyl-L-histidyl-L-tryptophyl-L-seryl-L-tyrosyl-3-(2-naphthyl)-D-alanyl-L-leucyl-L-arginyl-L-prolylglycinamide acetate salt hydrate

Empirical Formula (Hill Notation): C66H83N17O13 · xC2H4O2 · yH2O CAS号: 86220-42-0 分子量: 1322.47 (anhydrous free base basis) MDL编号: MFCD00895733 PubChem化学物质编号: 329818673 NACRES: NA.77
¥2,760.00

盐酸萘夫昔定,Nafoxidine hydrochloride;≥98% (HPLC)

PZ0118
别名:萘夫昔定盐酸盐;CP-5600;1-[2-[4-(3,4-二氢-6-甲氧基-2-苯基-1-萘基)苯氧基]乙基]吡咯烷盐酸盐;1-[2-[4-(3,4-dihydro-6-methoxy-2-phenyl-1-naphthalenyl)phenoxy]ethyl]-pyrrolidine hydrochloride, Nafoxidene hydrochloride, PNU-0011100

Empirical Formula (Hill Notation): C29H31NO2 · HCl CAS号: 1847-63-8 分子量: 462.02 MDL编号: MFCD00056572 PubChem化学物质编号: 329823710 NACRES: NA.77
¥1,412.50

NI-42,≥98% (HPLC)

PZ0348
别名:4-氰基-N-(1,2-二氢-1,3-二甲基-2-氧代-6-喹啉基)苯磺酰胺;4-Cyano-N-(1,2-dihydro-1,3-dimethyl-2-oxo-6-quinolinyl)benzenesulfonamide

Empirical Formula (Hill Notation): C18H15N3O3S CAS号: 1884640-99-6 分子量: 353.40 MDL编号: MFCD30290161
¥1,591.58

OSU6162盐酸盐,OSU6162 hydrochloride;≥98% (HPLC)

PZ0177
别名:PNU-96391;PNU-0096391;OSU-6162;(S)-(-)-(3-甲磺酰基苯基)-1-丙基哌啶盐酸盐;(S,S)-3-[3-(甲基磺酰基)苯基]-1-丙基哌啶盐酸盐;(S)-(-)-(3-methanesulfonyl-phenyl)-1-propyl-piperidine hydrochloride; (S,S)-3-[3-(Methylsulfonyl)phenyl]-1-propylpiperidine hydrochloride

Empirical Formula (Hill Notation): C15H23NO2S·HCl CAS号: 156907-84-5 分子量: 317.87 MDL编号: MFCD09753276 PubChem化学物质编号: 329823751 NACRES: NA.77
¥1,878.60

PD-156707,≥98% (HPLC)

PZ0141
别名:α-[2-(4-甲氧基苯基)-2-氧代-1-[(3,4,5-三甲氧基苯基)甲基]亚乙基]-1,3-苯并二氧戊环-5-乙酸钠盐;α-[2-(4-Methoxyphenyl)-2-oxo-1-[(3,4,5-trimethoxyphenyl)methyl]ethylidene]-1,3-benzodioxole-5-acetic acid sodium salt

Empirical Formula (Hill Notation): C28H25O9·Na CAS号: 162412-70-6 分子量: 528.48 PubChem化学物质编号: 329823726 NACRES: NA.77
¥1,763.90

PD161989 2-羟基乙烷磺酸酯,PD-161989 2-Hydroxyethanesulfonate,≥98% (HPLC)

PZ0144
别名:1,4-二氢-6-甲基-7-硝基-5-(1-吡咯烷甲基)-2,3-喹喔啉 2-羟基乙烷磺酸盐;1,4-Dihydro-6-methyl-7-nitro-5-(1-pyrrolodinemethyl)-2,3-quinoxaline 2-hydroxyethanesulfonic acid salt, PD-161989 isethionate salt, PD-161989 2-hydroxyethanesulfonic acid salt

Empirical Formula (Hill Notation): C14H16N4O4 · C2H6O4S CAS号: 186268-07-5 (free base) 分子量: 430.43 MDL编号: MFCD18452848 PubChem化学物质编号: 329823729 NACRES: NA.77
¥2,361.48

PD166285水合物,PD-166285 hydrate;≥98% (HPLC)

PZ0116
别名:6-(2,6-二氯苯基)-2-[[4-[2-(二乙氨基)乙氧基]苯基]氨基]-8-甲基吡啶并[2,3-d]嘧啶-7(8H)-酮二盐酸盐水合物;6-(2,6-Dichlorophenyl)-2-[[4-[2-(diethylamino)ethoxy]phenyl]amino]-8-methyl-pyrido[2,3-d]pyrimidin-7(8H)-one dihydrochloride hydrate

Empirical Formula (Hill Notation): C26H27Cl2N5O2·2HCl 分子量: 585.35 MDL编号: MFCD17215957 PubChem化学物质编号: 329823708 NACRES: NA.77
¥2,159.94

PD-85639,≥98% (HPLC)

PZ0370
别名:PD 85639, PD85,639, PD85639;N-[3-(2,6-二甲基-1-哌啶基)丙基]-α-苯基苯乙酰胺;N-[3-(2,6-Dimethyl-1-piperidinyl)propyl]-α-phenylbenzeneacetamide

Empirical Formula (Hill Notation): C24H32N2O CAS号: 149838-21-1 分子量: 364.52 MDL编号: MFCD14635427 NACRES: NA.77
¥1,641.30