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20,000多种特异性抑制剂、激动剂作用于表观遗传学、PI3K/Akt/mTOR、凋亡、MAPK、Wnt等20多个信号通路的375个靶点蛋白,覆盖癌症、神经科学、免疫学等热门疾病研究领域。BSZH北实纵横科学公司的50多种活性化合物库,包含10,000多种具有生物活性的小分子化合物,可用于高通量筛选 (HTS)和高内涵筛选 (HCS),是进行新药筛选和新适应症发现等研究的专业工具。
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3-AP,≥98% (HPLC)
SML0568
别名:[(3-氨基吡啶-2-基)亚甲基氨基]硫脲;3-Aminopyridine-2-carboxaldehyde thiosemicarbazone, 3-AP, PAN-811
Empirical Formula (Hill Notation): C7H9N5S CAS号: 143621-35-6 分子量: 195.24 NACRES: NA.77
Empirical Formula (Hill Notation): C7H9N5S CAS号: 143621-35-6 分子量: 195.24 NACRES: NA.77
¥907.39
ITSA-1,≥98% (HPLC), solid
I4159
别名:1-(2,4-二氯苯甲酰基)-1H-苯并三唑;1-(2,4-Dichlorobenzoyl)-1H-benzotriazole, Inhibitor-1 of Trichostatin A, N-(1H-Benzotriazol-1-yl)-2,4-dichlorobenzamide
Empirical Formula (Hill Notation): C13H7Cl2N3O CAS号: 200626-61-5 分子量: 292.12 MDL编号: MFCD00195103 PubChem化学物质编号: 24724515
Empirical Formula (Hill Notation): C13H7Cl2N3O CAS号: 200626-61-5 分子量: 292.12 MDL编号: MFCD00195103 PubChem化学物质编号: 24724515
¥1,726.00
Madrasin,≥98% (HPLC)
SML1409
别名:RNA剪接抑制剂;2-[((7-甲氧基-4-甲基-2-喹唑啉基)氨基] -5,6-二甲基-4(1H)-嘧啶酮(9CI);2-(7-甲氧基-4-甲基-喹唑啉-2-基氨基)-5,6-二甲基-3H-嘧啶-4-酮, 4(1H)-嘧啶酮,2-[((7-甲氧基-4-甲基-2-喹唑啉基)氨基] -5,6-二甲基-(9CI), 4(3H)-嘧啶酮,2-[((7-甲氧基-4-甲基-2-喹唑啉基)氨基] -5,6-二甲基-, DDD00107587;2-(7-Methoxy-4-methyl-quinazolin-2-ylamino)-5,6-dimethyl-3H-pyrimidin-4-one, 2-[(7-Methoxy-4-methyl-2-quinazolinyl)amino]-5,6-dimethyl-4(1H)-pyrimidinone (9CI), 4(1H)-Pyrimidinone, 2-[(7-methoxy-4-methyl-2-quinazolinyl)amino]-5,6-dimethyl-(9CI), 4(3H)-Pyrimidinone, 2-[(7-methoxy-4-methyl-2-quinazolinyl)amino]-5,6-dimethyl-, DDD00107587, RNAsplicing inhibitor
Empirical Formula (Hill Notation): C16H17N5O2 CAS号: 374913-63-0 分子量: 311.34 MDL编号: MFCD02233199 PubChem化学物质编号: 329825856
Empirical Formula (Hill Notation): C16H17N5O2 CAS号: 374913-63-0 分子量: 311.34 MDL编号: MFCD02233199 PubChem化学物质编号: 329825856
¥1,364.05
MC1568;≥99% (HPLC)
S06080
别名:3- [5-(3-(3-氟苯基)-3-氧代丙烯-1-基)-1-甲基-1H-吡咯-2-基]-N-羟基-2-丙烯酰胺;3-[5-(3-(3-Fluorophenyl)-3-oxopropen-1-yl)-1-methyl-1H-pyrrol-2-yl]-N-hydroxy-2-propenamide
Empirical Formula (Hill Notation): C17H15FN2O3 CAS号: 852475-26-4 分子量: 314.31 PubChem化学物质编号: 329817891
Empirical Formula (Hill Notation): C17H15FN2O3 CAS号: 852475-26-4 分子量: 314.31 PubChem化学物质编号: 329817891
¥1,943.60
Sapanisertib [INK128, MLN0128];≥99% (HPLC)
S06075
别名:5-(4-氨基-1-异丙基-1H-吡唑并[3,4-d]嘧啶-3-基)苯并[d]恶唑-2-胺;沙帕色替;INK-128;3-(2-amino-5-benzoxazolyl)-1-(1-methylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
CAS:1224844-38-5;分子式:C15H15N7O;分子量:309.33;MDL:MFCD22124893
CAS:1224844-38-5;分子式:C15H15N7O;分子量:309.33;MDL:MFCD22124893
¥1,750.00
SB939 [Pracinostat];≥99% (HPLC)
S06081
别名:(E)-3-(2-丁基-1-(2-(二乙氨基)乙基)-1H-苯并[d]咪唑-5-基)-N-羟基丙烯酰胺;(E)-3-(2-Butyl-1-(2-(diethylamino)ethyl)-1H-benzo[d]imidazol-5-yl)-N-hydroxyacrylamide
CAS:929016-96-6;分子式:C20H30N4O2;分子量:358.48
CAS:929016-96-6;分子式:C20H30N4O2;分子量:358.48
¥1,260.00
YK-4-279;≥99% (HPLC)
S06076
别名:4,7-二氯-3-羟基-3-(2(4-甲氧基苯基)-2-氧代乙基)二氢吲哚-2-酮;4,7-Dichloro-1,3-dihydro-3-hydroxy-3-[2-(4-methoxyphenyl)-2-oxoethyl]-2H-indol-2-one
CAS:1037184-44-3;分子式:C17H13Cl2NO4;分子量:366.20;MDL:MFCD18382120
CAS:1037184-44-3;分子式:C17H13Cl2NO4;分子量:366.20;MDL:MFCD18382120
¥976.00
西他司他,Citarinostat [ACY-241];≥99% (HPLC)
S06078
别名:HDAC-IN-2;2-(2-氯苯基)(苯基)氨基)-N-(7-羟基氨基)-7-氧代庚基)嘧啶-5-甲酰胺;2-((2-chlorophenyl)(phenyl)amino)-N-(7-(hydroxyamino)-7-oxoheptyl)pyrimidine-5-carboxamide
CAS:1316215-12-9;分子式:C24H26ClN5O3;分子量:467.95
CAS:1316215-12-9;分子式:C24H26ClN5O3;分子量:467.95
¥1,950.00
CI−994,≥98% (HPLC), powder
C0621
别名:4-乙酰氨基-N-(2′-氨基苯基)苯甲酰胺;乙酰地那林;醋地那林;4-Acetylamino-N-(2′-aminophenyl)benzamide, Acetyldinaline, Tacedinaline
Empirical Formula (Hill Notation): C15H15N3O2 CAS号: 112522-64-2 分子量: 269.30 MDL编号: MFCD00866266 PubChem化学物质编号: 329774808 NACRES: NA.77
Empirical Formula (Hill Notation): C15H15N3O2 CAS号: 112522-64-2 分子量: 269.30 MDL编号: MFCD00866266 PubChem化学物质编号: 329774808 NACRES: NA.77
¥1,473.31
DS16570511,≥99.0%
HY-115595
DS16570511 是一种细胞渗透性的线粒体钙单核转运蛋白 (mitochondrial calcium uniporter) 抑制剂,阻断了依赖于 MCU 或 MICU1 的 Ca2+ 流入增加。
¥1,760.00
AP20187,≥98% (HPLC)
SML2838
别名:蛋白质二聚化的化学诱导剂;(2S,2′S)-1-[(2S)-1-oxo-2-(3,4,5-trimethoxyphenyl)butyl]-2-piperidinecarboxylic acid, 2,2′-[[2-[(dimethylamino)methyl]-1,3-propanediyl]bis[imino(2-oxo-2,1-ethanediyl)oxy-3,1-phenylene[(1R)-3-(3,4-dimethoxyphenyl)propylidene]]] ester
Empirical Formula (Hill Notation): C82H107N5O20 CAS号: 195514-80-8 分子量: 1482.75 MDL编号: MFCD28167729
Empirical Formula (Hill Notation): C82H107N5O20 CAS号: 195514-80-8 分子量: 1482.75 MDL编号: MFCD28167729
¥1,306.87
AP20187,≥99.5% (HPLC)
HY-13992
别名:蛋白质二聚化的化学诱导剂;(2S,2′S)-1-[(2S)-1-oxo-2-(3,4,5-trimethoxyphenyl)butyl]-2-piperidinecarboxylic acid, 2,2′-[[2-[(dimethylamino)methyl]-1,3-propanediyl]bis[imino(2-oxo-2,1-ethanediyl)oxy-3,1-phenylene[(1R)-3-(3,4-dimethoxyphenyl)propylidene]]] ester
Empirical Formula (Hill Notation): C82H107N5O20 CAS号: 195514-80-8 分子量: 1482.75 MDL编号: MFCD28167729
Empirical Formula (Hill Notation): C82H107N5O20 CAS号: 195514-80-8 分子量: 1482.75 MDL编号: MFCD28167729
¥4,360.00