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信号通路, 信号转导, Cell Signaling

20,000多种特异性抑制剂、激动剂作用于表观遗传学、PI3K/Akt/mTOR、凋亡、MAPK、Wnt等20多个信号通路的375个靶点蛋白,覆盖癌症、神经科学、免疫学等热门疾病研究领域。BSZH北实纵横科学公司的50多种活性化合物库,包含10,000多种具有生物活性的小分子化合物,可用于高通量筛选 (HTS)和高内涵筛选 (HCS),是进行新药筛选和新适应症发现等研究的专业工具。

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PF-02413873,≥98% (HPLC)

PZ0367
别名:4-[3-环丙基-1-甲砜基甲基-5-甲基吡唑-4-基]氧基-2,6-二甲基苯腈;4-[[3-环丙基-5-甲基-1-[(甲基磺酰基)甲基]-1H-吡唑-4-基]氧基]-2,6-二甲基苯腈;4-3-Cyclopropyl-1-(mesylmethyl)-5-methyl-1H-pyrazol-4-yloxy-2,6-dimethylbenzonitrile, PF 2413873, PF-2413873, 4-3-Cyclopropyl-5-methyl-1-(methylsulfonyl)methyl-1H-pyrazol-4-yloxy-2,6-dimethyl-benzonitrile

Empirical Formula (Hill Notation): C18H21N3O3S CAS号: 936345-35-6 分子量: 359.44 MDL编号: MFCD16987601 NACRES: NA.77
¥1,563.33

PF-06273340,≥98% (HPLC)

PZ0254
别名:N-(5-{2-Amino-7-(2-hydroxy-1 ,1-dimethylethyl)-7H-pyrrolo2,3-dpyrimidin-5- ylcarbonyl}pyridin-3-yl)-2-(5-chloropyridin-2-yl)acetamide, PF 06273340, N-5-2-Amino-7-(2-hydroxy-1,1-dimethylethyl)-7H-pyrrolo2,3-dpyrimidin-5-ylcarbonyl-3-pyridinyl-5-chloro-2-pyridineacetamide, PF06273340

Empirical Formula (Hill Notation): C23H22ClN7O3 CAS号: 1402438-74-7 分子量: 479.92 PubChem化学物质编号: 329823793 NACRES: NA.77
¥1,391.58

甲磺酸地拉韦啶,Delavirdine mesylate;≥98% (HPLC)

PZ0180
别名:地拉夫定甲磺酸盐;Rescriptor;N-[2-[[4-[3-[(1-甲基乙基)氨基]-2-吡啶基]-1-哌嗪基]羰基]-1H-吲哚-5-基]甲磺酰胺甲磺酸酯;N-2-4-3-(1-Methylethyl)amino-2-pyridinyl-1-piperazinylcarbonyl-1H-indol-5-ylmethanesulfonamide mesylate

Empirical Formula (Hill Notation): C22H28N6O3S · CH3SO3H CAS号: 147221-93-0 分子量: 552.67 MDL编号: MFCD00866948 PubChem化学物质编号: 329823754 NACRES: NA.77
¥1,378.60

PF-06282999,≥98% (HPLC)

PZ0375
别名:PF 06282999, PF06282999;2-(6-(5-氯-2-甲氧基苯基)-4-氧代-2-硫代-3,4-二氢嘧啶-1(2H)-基)乙酰胺;6-(5-氯-2-甲氧基苯基)-3,4-二氢-4-氧代-2-硫代-1(2H)-嘧啶乙酰胺;2-(6-(5-Chloro-2-methoxyphenyl)-4-oxo-2-thioxo-3,4-dihydropyrimidin-1(2H)-yl)acetamide, 6-(5-Chloro-2-methoxyphenyl)-3,4-dihydro-4-oxo-2-thioxo-1(2H)-pyrimidineacetamide

Empirical Formula (Hill Notation): C13H12ClN3O3S CAS号: 1435467-37-0 分子量: 325.77 MDL编号: MFCD30533689 NACRES: NA.77
¥1,281.78

PF4800567盐酸盐,PF-4800567 hydrochloride;≥98% (HPLC)

PZ0328
别名:PF4800567 HCl;3-[(3-氯苯氧基)甲基]-1-(四氢-2H-吡喃-4-基)-1H-吡唑并[3,4-d]嘧啶-4-胺盐酸盐;3-(3-Chlorophenoxy)methyl-1-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo3,4-dpyrimidin-4-amine hydrochloride, PF 4800567

Empirical Formula (Hill Notation): C17H18ClN5O2 · HCl CAS号: 1391052-28-0 分子量: 396.27
¥1,591.58

CP154526盐酸盐,CP-154526 hydrochloride;≥98% (HPLC)

PZ0100
别名:N-丁基-N-乙基-2,5-二甲基-7-(2,4,6-三甲基苯基)-7H-吡咯并[2,3-d]嘧啶-4-胺单盐酸盐;N-Butyl-N-ethyl-2,5-dimethyl-7-(2,4,6-trimethylphenyl)-7H-pyrrolo2,3-dpyrimidin-4-amine monohydrochloride

Empirical Formula (Hill Notation): C23H32N4 · HCl CAS号: 257639-98-8 分子量: 400.99 MDL编号: MFCD07364047 PubChem化学物质编号: 329823693 NACRES: NA.77
¥1,720.40

PD-180970,≥98% (HPLC)

PZ0142
别名:6-(2,6-二氯苯基)-2-(4-氟-3-甲基苯基)氨基]-8-甲基吡啶并[2,3-d]嘧啶-7(8H)酮;6-(2,6-Dichlorophenyl)-2-(4-fluoro-3-methylphenyl)amino-8-methyl-pyrido2,3-dpyrimidin-7(8H)-one, PF-1515965

Empirical Formula (Hill Notation): C21H15Cl2FN4O CAS号: 287204-45-9 分子量: 429.27 MDL编号: MFCD10565929 PubChem化学物质编号: 329823727 NACRES: NA.77
¥1,754.46

WAY-362450,≥98% (HPLC)

PZ0267
别名:WAY362450;XL335;异氟硼酸异丙酯, 3-(3,4-二氟-苯甲酰基)-1,1-二亚甲基-1,2,3,6-四氢-阿斯皮诺4,5-b吲哚-5-羧酸异丙酯, FXR 450, WAY 362450, 3-(3,4-二氟苯甲酰基)-1,2,3,6-四氢-1,1-二甲基-氮杂环庚烷4,5-b吲哚-5-羧酸1-甲基乙基酯;Turofexorate isopropyl, 3-(3,4-Difluorobenzoyl)-1,2,3,6-tetrahydro-1,1-dimethyl-azepino4,5-bindole-5-carboxylic acid 1-methylethyl ester, XL335, 3-(3,4-Difluoro-benzoyl)-1,1-dimethylene-1,2,3,6-tetrahydro-azepino 4,5-bindole-5-carboxylic acid isopropyl ester, FXR 450

Empirical Formula (Hill Notation): C25H24F2N2O3 CAS号: 629664-81-9 分子量: 438.47 MDL编号: MFCD13181507 PubChem化学物质编号: 329823801
¥1,091.58

PD-184161,≥98% (HPLC)

PZ0112
别名:PD184161;UK-287074;5-溴-2-[(2-氯-4-碘苯基)氨基]-N-环丙基甲氧基-3,4-二氟苯甲酰胺;5-Bromo-2-(2-chloro-4-iodophenyl)amino-N-(cyclopropylmethoxy)-3,4-difluoro-benzamide, PF-1529483, PF-3011370

Empirical Formula (Hill Notation): C17H13BrClF2IN2O2 CAS号: 212631-67-9 分子量: 557.56 MDL编号: MFCD16038897 PubChem化学物质编号: 329823704
¥1,378.60

PF-04885614,≥98% (HPLC)

PZ0210
别名:PF04885614;1-甲基-1-[4-(4-三氟甲氧基苯基)-1H-咪唑-2-基]乙胺;1-Methyl-1-4-(4-trifluoromethoxy-phenyl)-1H-imidazol-2-yl-ethylamine

Empirical Formula (Hill Notation): C13H14F3N3O 分子量: 285.26 NACRES: NA.77
¥1,104.01

(S)-PFI-2;≥98% (HPLC)

PZ0312
别名:PF-06477717盐酸盐;PF06477717;(R)-8-氟-N-(1-氧代-1-(吡咯烷-1-基)-3-(3-(三氟甲基)苯基)丙-2-基)-1,2,3,4-四氢异喹啉-6磺酰胺 盐酸盐, (S)-PFI-2 盐酸盐;(S)-8-Fluoro-N-(1-oxo-1-(pyrrolidin-1-yl)-3-(3-(trifluoromethyl)phenyl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide hydrochloride, PF-06477717 hydrochloride, (S)-PFI-2 hydrochloride

Empirical Formula (Hill Notation): C23H25F4N3O3S · HCl CAS号: 1627607-88-8 分子量: 535.98 PubChem化学物质编号: 329823832 NACRES: NA.77
¥1,591.58

PF-03814735,≥98% (HPLC)

PZ0218
别名:N-[2-[(1S,4R)-6-[[4-(环丁基氨基)-5-(三氟甲基)-2-嘧啶基]氨基]-1,2,3,4-四氢萘-1,4-亚胺-9-基]-2-氧代乙基]-乙酰胺;N-[2-[(1S,4R)-6-[[4-(Cyclobutylamino)-5-(trifluoromethyl)-2-pyrimidinyl]amino]-1,2,3,4-tetrahydronaphthalen-1,4-imin-9-yl]-2-oxoethyl]-acetamide

Empirical Formula (Hill Notation): C23H25F3N6O2 CAS号: 942487-16-3 分子量: 474.48 NACRES: NA.77
¥1,591.58