常用生化试剂, Core BioReagents
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妥卡替尼,Irbinitinib [ARRY-380];≥99% (HPLC)
S06227
别名:Tucatinib;ONT 380;N6-(4,4-Dimethyl-4,5-dihydrooxazol-2-yl)-N4-(3-methyl-4-((1,2,4)triazolo(1,5-a)pyridin-7-yloxy)phenyl)quinazoline-4,6-diamine
CAS:937263-43-9;分子式:C26H24N8O2;分子量:480.53
CAS:937263-43-9;分子式:C26H24N8O2;分子量:480.53
¥1,550.00
奥莫替尼 ,Olmutinib;≥99% (HPLC)
S06228
别名:HM 61713;BI1482694;N-(3-((2-((4-(4-甲基哌嗪-1-基)苯基)氨基)噻吩并[3,2-d]嘧啶-4-基)氧基)苯基)丙烯酰胺;N-{3-[(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}thieno[3,2-d]pyrimidin-4-yl)oxy]phenyl}prop-2-enamide
CAS:1353550-13-6;分子式:C26H26N6O2S;分子量:486.59
CAS:1353550-13-6;分子式:C26H26N6O2S;分子量:486.59
¥926.00
酪氨酸激酶抑制剂AG490,Tyrphostin AG 490;≥98% (HPLC)
T3434
别名:酪磷蛋白AG490;酪氨酸磷酸化抑制剂AG 490;2-氰基-3-(3,4-二羟基苯基)-N-(苄基)-2-丙烯酰胺, 2-氰基-3-(3,4-二羟基苯基)-N-(苯甲基)-2-丙烯酰胺;2-Cyano-3-(3,4-dihydroxyphenyl)-N-(benzyl)-2-propenamide, 2-Cyano-3-(3,4-dihydroxyphenyl)-N-(phenylmethyl)-2-propenamide
Empirical Formula (Hill Notation): C17H14N2O3 CAS号: 133550-30-8 分子量: 294.30 MDL编号: MFCD00236452 PubChem化学物质编号: 24278732 NACRES: NA.77
Empirical Formula (Hill Notation): C17H14N2O3 CAS号: 133550-30-8 分子量: 294.30 MDL编号: MFCD00236452 PubChem化学物质编号: 24278732 NACRES: NA.77
¥1,107.45
Defactinib,[VS-6063, PF-04554878];≥99% (HPLC)
D06230
别名:VS-6063;PF-04554878;N-methyl-4-((4-(((3-(N-methylmethylsulfonamido)pyrazin-2-yl)methyl)amino)-5-(trifluoromethyl)pyrimidin-2-yl)amino)benzamide
CAS:1345713-71-4;分子式:C20H21F3N8O3S;分子量:510.49
CAS:1345713-71-4;分子式:C20H21F3N8O3S;分子量:510.49
¥1,550.00
PF431396水合物,PF-431396 hydrate;≥98% (HPLC)
PZ0185
别名:N-甲基-N-(2-(((2-((2-氧代二氢吲哚-5-基)氨基)-5-(三氟甲基)嘧啶-4-基)氨基)甲基)苯基)甲磺酰胺;N-[2-[[[2-[(2,3-dihydro-2-oxo-1H-indol-5-yl)amino]-5-(trifluoromethyl)-4-pyrimidinyl]amino]methyl]phenyl]-N-methyl-Methanesulfonamide hydrate
Empirical Formula (Hill Notation): C22H21F3N6O3S · xH2O CAS号: 717906-29-1 分子量: 506.50 (anhydrous basis) MDL编号: MFCD21608515 PubChem化学物质编号: 329823759 NACRES: NA.77
Empirical Formula (Hill Notation): C22H21F3N6O3S · xH2O CAS号: 717906-29-1 分子量: 506.50 (anhydrous basis) MDL编号: MFCD21608515 PubChem化学物质编号: 329823759 NACRES: NA.77
¥1,175.20
FIIN-2,≥99% (HPLC)
F06232
别名:FGFR抑制剂;FIIN2;FIIN 2;N-(4-(3,5-二甲氧基苯基)-7-(4-(4-甲基哌嗪-1-基)苯基)氨基)-2-氧代-3,4-二氢嘧啶并[4,5-d]嘧啶-1(2H)-甲基)苯基)丙烯酰胺;N-(4-((3-(3,5-dimethoxyphenyl)-7-((4-(4-methylpiperazin-1-yl)phenyl)amino)-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2H)-yl)methyl)phenyl)acrylamide
CAS:1633044-56-0;分子式:C35H38N8O4;分子量:634.73
CAS:1633044-56-0;分子式:C35H38N8O4;分子量:634.73
¥1,830.00
Infigratinib,[BGJ398, NVP-BGJ398];≥99% (HPLC)
B06233
别名:3-(2,6-二氯-3,5-二甲氧基苯基)-1-[6-[[4-(4-乙基哌嗪-1-基)苯基]氨基]嘧啶-4-基]-1-甲基脲;3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-[6-[4-(4-ethylpiperazin-1-yl)anilino]pyrimidin-4-yl]-1-methylurea
CAS:872511-34-7;分子式:C26H31Cl2N7O3;分子量:560.47;MDL:MFCD22123241
CAS:872511-34-7;分子式:C26H31Cl2N7O3;分子量:560.47;MDL:MFCD22123241
¥962.00
PD-166866,≥98% (HPLC)
PZ0114
别名:1-(2-氨基-6-(3,5-二甲氧基苯基)吡啶并[2,3-d]嘧啶-7-基)-3-(叔丁基)脲;PD166866;PD 166866;1-[2-Amino-6-(3,5-dimethoxyphenyl)-pyrido[2,3-d]pyrimidin-7-yl]-3-tert-butyl urea
Empirical Formula (Hill Notation): C20H24N6O3 CAS号: 192705-79-6 分子量: 396.44 MDL编号: MFCD12922514 PubChem化学物质编号: 329823706 NACRES: NA.77
Empirical Formula (Hill Notation): C20H24N6O3 CAS号: 192705-79-6 分子量: 396.44 MDL编号: MFCD12922514 PubChem化学物质编号: 329823706 NACRES: NA.77
¥1,220.40
UNC2025,≥99% (HPLC)
U06235
别名:UNC-2025;UNC2025 2HCl;(1r,4r)-4-(2-(butylamino)-5-(4-((4-methylpiperazin-1-yl)methyl)phenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)cyclohexanol;反式-4-(2-(丁胺基)-5-(4-((4-甲基哌嗪-1-基)甲基)苯基)-7H-吡咯并[2,3-d]嘧啶-7-基)环己醇
CAS:1429881-91-3;分子式:C28H40N6O;分子量:476.66
CAS:1429881-91-3;分子式:C28H40N6O;分子量:476.66
¥1,732.00
NT157 [NT-157],≥99% (HPLC)
N06236
别名:(2E)-3-(3-Bromo-4,5-dihydroxyphenyl)-N-[(3,4,5-trihydroxyphenyl)methyl]-2-propenethioamide;(E)-3-(3-Bromo-4,5-dihydroxyphenyl)-n-(3,4,5-trihydroxybenzyl)prop-2-enethioamide
CAS:1384426-12-3;分子式:C16H14BrNO5S;分子量:412.25
CAS:1384426-12-3;分子式:C16H14BrNO5S;分子量:412.25
¥1,550.00
IRAK-1/4抑制剂I,IRAK-1/4 Inhibitor I;≥98% (HPLC), solid
I5409
别名:1-(2-(4-吗啉基)乙基)-2-(3-硝基苯甲酰基)苯并咪唑, N-(2-吗啉基乙基)-2-(3-硝基苯甲酰胺)-苯并咪唑;1-(2-(4-Morpholinyl)ethyl)-2-(3-nitrobenzoylamino)benzimidazole, N-(2-Morpholinylethyl)-2-(3-nitrobenzoylamido)-benzimidazole
Empirical Formula (Hill Notation): C20H21N5O4 分子量: 395.41 MDL编号: MFCD09752602 PubChem化学物质编号: 329815384 NACRES: NA.77
Empirical Formula (Hill Notation): C20H21N5O4 分子量: 395.41 MDL编号: MFCD09752602 PubChem化学物质编号: 329815384 NACRES: NA.77
¥2,196.46
AG 1296,≥98% (HPLC)
658551
别名:AG-1296;AG1296;6,7-Dimethoxy-3-phenylquinoxaline;6,7-二甲氧基-2-苯基喹喔啉
Empirical Formula (Hill Notation): C16H14N2O2 CAS号: 146535-11-7 分子量: 266.29 MDL编号: MFCD00270913
Empirical Formula (Hill Notation): C16H14N2O2 CAS号: 146535-11-7 分子量: 266.29 MDL编号: MFCD00270913
¥1,950.00