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信号通路, 信号转导, Cell Signaling

20,000多种特异性抑制剂、激动剂作用于表观遗传学、PI3K/Akt/mTOR、凋亡、MAPK、Wnt等20多个信号通路的375个靶点蛋白,覆盖癌症、神经科学、免疫学等热门疾病研究领域。BSZH北实纵横科学公司的50多种活性化合物库,包含10,000多种具有生物活性的小分子化合物,可用于高通量筛选 (HTS)和高内涵筛选 (HCS),是进行新药筛选和新适应症发现等研究的专业工具。

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放线菌素D [更生霉素],Actinomycin D;from Streptomyces sp., ≥95% (HPLC)

A4262
别名:放线菌素 C1;放线菌素 IV;D放线菌素;Actinomycin C1, Actinomycin IV, Dactinomycin

Empirical Formula (Hill Notation): C62H86N12O16 CAS号: 50-76-0 分子量: 1255.42 Beilstein: 605235 EC 号: 200-063-6 MDL编号: MFCD00005033 PubChem化学物质编号: 24890842 NACRES: NA.76
¥1,854.00

放线菌素D [更生霉素],Actinomycin D;from Streptomyces sp., suitable for cell culture, ≥95%

A9415
别名:放线菌素 C1;放线菌素 IV;D放线菌素;Actinomycin C1, Actinomycin IV, Dactinomycin

Empirical Formula (Hill Notation): C62H86N12O16 CAS号: 50-76-0 分子量: 1255.42 Beilstein: 605235 EC 号: 200-063-6 MDL编号: MFCD00005033 PubChem化学物质编号: 24891447 NACRES: NA.76
¥1,750.00

盐酸依达比星,Idarubicin hydrochloride [DMDR, IMI-30, Idamycin];pharmaceutical secondary standard, certified reference material

PHR2704
别名:依达比星盐酸盐标准品;(7S-cis)-9-Acetyl-7-[(3-amino-2,3,6-trideoxy-α-L-lyxo-hexopyranosyl)oxy]-7,8,9,10-tetrahydro-6,9,11-trihydroxy-5,12-naphthacenedione, 4-Demethoxydaunorubicin hydrochloride, DMDR, IMI-30, Idamycin

Empirical Formula (Hill Notation): C26H27NO9 · HCl CAS号: 57852-57-0 分子量: 533.95 MDL编号: MFCD00866457
¥6,750.00

盐酸依达比星,Idarubicin hydrochloride [DMDR, IMI-30, Idamycin];solid

I1656
别名:依达比星盐酸盐;(7S-cis)-9-Acetyl-7-[(3-amino-2,3,6-trideoxy-α-L-lyxo-hexopyranosyl)oxy]-7,8,9,10-tetrahydro-6,9,11-trihydroxy-5,12-naphthacenedione, 4-Demethoxydaunorubicin hydrochloride, DMDR, IMI-30, Idamycin

Empirical Formula (Hill Notation): C26H27NO9 · HCl CAS号: 57852-57-0 分子量: 533.95 EC 号: 260-990-7 MDL编号: MFCD00866457 PubChem化学物质编号: 24278488 NACRES: NA.77
¥976.00

利福布汀,Rifabutin;>98% (HPLC), powder

R3530
别名:利福布丁;安沙霉素;安沙地平;Ansamycin, Ansatipine (Farmitalia), LM-427, Mycobutin (Farmitalia)

Empirical Formula (Hill Notation): C46H62N4O11 CAS号: 72559-06-9 分子量: 847.00 NACRES: NA.77
¥1,350.00

利福布汀,Rifabutin;Pharmaceutical Secondary Standard; Certified Reference Material

PHR2611
别名:利福布汀标准品;利福布丁;安沙霉素;安沙地平;Ansamycin, Ansatipine (Farmitalia), LM-427, Mycobutin (Farmitalia)

Empirical Formula (Hill Notation): C46H62N4O11 CAS号: 72559-06-9 分子量: 847.00
¥2,660.00

格尔德霉素,Geldanamycin from Streptomyces hygroscopicus;≥98% (HPLC), powder

G3381
格尔德菌素;NSC 122750; Empirical Formula (Hill Notation): C29H40N2O9 CAS号: 30562-34-6 分子量: 560.64 MDL编号: MFCD00274570 PubChem化学物质编号: 329799914 NACRES: NA.77
¥4,650.00

17-烯丙基胺格尔德霉素,17-(Allylamino)-17-demethoxygeldanamycin [17-AAG];≥98% (HPLC), solid

A8476
别名:坦螺旋霉素;替拉替尼;17-(Allylamino)geldanamycin, 17-Demethoxy-17-allylamino geldanamycin, 17-AAG, CP 127374, Geldanamycin,17-demethoxy-17-(2-propenylamino)-, NSC 330507, Tanespimycin

Empirical Formula (Hill Notation): C31H43N3O8 CAS号: 75747-14-7 分子量: 585.69 MDL编号: MFCD04973892 PubChem化学物质编号: 329770957 NACRES: NA.77
¥2,650.00

人内皮抑素,Endostatin human;recombinant, expressed in E. coli, ≥98% (SDS-PAGE), ≥98% (HPLC), suitable for cell culture

SRP3031
内皮抑素是一种肿瘤血管生成抑制剂,属新一代抗肿瘤药物;NACRES NA.32
¥3,350.00

烟曲霉素,Fumagillin from Aspergillus fumigatus;≥90%, powder

F6771
别名: Fugillin Empirical Formula (Hill Notation): C26H34O7 CAS号: 23110-15-8 分子量: 458.54 EC 号: 245-433-8 MDL编号: MFCD03990453 PubChem化学物质编号: 24894920
¥1,750.00

人血管抑素K1-3,Angiostatin K1-3 human;≥90% (SDS-PAGE), recombinant, expressed in Pichia pastoris (without N-linked glycosylation)

A1477
第一个内源性肿瘤血管生成抑制因子,能直接特异地作用于血管内皮细胞、抑制其增殖、减少肿瘤血管生成;MDL number MFCD02685909
¥5,650.00

小鼠内皮抑素,Endostatin murine;recombinant, expressed in Pichia pastoris, ≥95% (SDS-PAGE)

E8279
内皮抑素是一种肿瘤血管生成抑制剂,新一代抗肿瘤药物;MDL number MFCD01866296
¥4,950.00